scanUNIQUE Delta Set RB

87 Kinases You Can’t Get From The Next Leading Provider

When it comes to kinase selectivity and off-target profiling, kinase panel size matters! Larger panels provide not only a better measure of compound selectivity, but a more comprehensive view of potential off-target activity that smaller panels may overlook.

See for yourself how KINOMEscan compares to the competition using our scanUNIQUE Delta Set panels, or contact us to receive more information about the assays missing in your current solution provider's portfolio. Then request a quote to see what you're missing!
 

Panel Highlights and Benefits

  • 87 kinases not available from the next leading provider
  • Comprehensive view of potential off-target activity that smaller panels may overlook
  • Avoid costly decisions or even lost opportunities due to incomplete data

 

Delta Set Rb
Red circles represent unique KINOMEscan™ kinases not currently available from the next leading provider.

Case Study: Assessing Compound Selectivity & Potency Across Delta Set RB Assays

 

Sunitinib


Sunitinib

Erlotinib


Erlotinib

Dasatinib


Dasatinib
Kd values < 3 µM for three FDA-approved kinase inhibitors across the 87 kinases not available from the next leading provider.

 

scanUNIQUE™, Delta Set RB - 87 Kinases
AAK1ACVR2AACVR2BADCK3ADCK4ANKK1ASK2BIKE
BMPR1ABUB1CAMK4CASKCDC2L1CDC2L2CDC2L5CDK11
CDK8CDKL1CDKL2CDKL3CDKL5CITCSNK1A1LDCAMKL3
DMPK2DRAK2EPHB6ERBB3ERK3ERK4ERK5ERK8
ERN1GAKHPK1HUNKICKIRAK3LATS1LIMK2
LZKMAKMAP3K15MAP3K4MAP4K3MAST1MEK3MEK5
MKK7MYLK4MYO3ANEK5NIM1PCTK1PCTK2PCTK3
PFTAIRE2PFTK1PIK3C2BPIK3C2GPIK4CBPIP5K1APIP5K1CPIP5K2B
PIP5K2CPKMYT1PRP4QSKRIOK1RIOK2RIOK3RIPK1
RIPK4SBK1SgK110SNRKSTK35STK36TESK1TIE1
TNNI3KTRPM6WEE2YANK1YANK2YANK3YSK4