ACVR1
KINASE INFORMATION
Kinase Name
activin A receptor, type I
Entrez Gene Symbol
ACVR1
Entrez Gene ID
90
Aliases
ACTRI; ACVR1; ACVR1A; ACVRLK2; ALK2; FOP; SKR1; TSRI
Kinase Group
TKL
Species
Human
PROTEIN INFORMATION
Accession #
NP_001096.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.69
Panel
Delta Set CA; Delta Set CE; Delta Set M; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
75 nM
Dasatinib
620 nM
JNJ-7706621
5900 nM