ACVRL1
KINASE INFORMATION
Kinase Name
activin A receptor type II-like 1
Entrez Gene Symbol
ACVRL1
Entrez Gene ID
94
Aliases
ACVRL1; ACVRLK1; ALK1; ALK-1; HHT; HHT2; ORW2; SKR3; TSR-I
Kinase Group
TKL
Species
Human
PROTEIN INFORMATION
Accession #
NP_000011.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.64
Panel
Delta Set CA; Delta Set CE; Delta Set I; Delta Set M; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
2200 nM
Dasatinib
460 nM
JNJ-7706621
2900 nM