ALK
KINASE INFORMATION
Kinase Name
anaplastic lymphoma receptor tyrosine kinase
Entrez Gene Symbol
ALK
Entrez Gene ID
238
Aliases
ALK; CD246; NBLST3; TFG/ALK
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_004295.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.66
Panel
Delta Set I; scanEDGE; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
PKC-412
270 nM
Staurosporine
32 nM
Sunitinib
170 nM