AMPK-alpha2
KINASE INFORMATION
Kinase Name
protein kinase, AMP-activated, alpha 2 catalytic subunit
Entrez Gene Symbol
PRKAA2
Entrez Gene ID
5563
Aliases
AMPK; AMPK2; AMPKa2; AMPK-alpha2; PRKAA; PRKAA2
Kinase Group
CAMK
Species
Human
PROTEIN INFORMATION
Accession #
NP_006243.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.75
Panel
Delta Set CE; Delta Set M; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
PKC-412
460 nM
SU-14813
290 nM
Sunitinib
89 nM