ANKK1
KINASE INFORMATION
Kinase Name
ankyrin repeat and kinase domain containing 1
Entrez Gene Symbol
ANKK1
Entrez Gene ID
255239
Aliases
ANKK1; PKK2; SgK288
Kinase Group
TKL
Species
Human
PROTEIN INFORMATION
Accession #
NP_848605.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.75
Panel
Delta Set CA; Delta Set CE; Delta Set I; Delta Set M; Delta Set RB; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CHIR-258/TKI-258
79 nM
SU-14813
160 nM
Sunitinib
310 nM