AXL
KINASE INFORMATION
Kinase Name
AXL receptor tyrosine kinase
Entrez Gene Symbol
AXL
Entrez Gene ID
558
Aliases
AXL; JTK11; UFO
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_001690.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.74
Panel
scanEDGE; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
35 nM
Staurosporine
6.8 nM
Sunitinib
9 nM
ZD-6474
250 nM