BIKE
KINASE INFORMATION
Kinase Name
BMP2 inducible kinase
Entrez Gene Symbol
BMP2K
Entrez Gene ID
55589
Aliases
BIKE; BMP2K; DKFZp434K0614; DKFZp434P0116; HRIHFB2017
Kinase Group
Other
Species
Human
PROTEIN INFORMATION
Accession #
NP_060063.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.6
Panel
Delta Set CA; Delta Set CE; Delta Set I; Delta Set M; Delta Set RB; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CHIR-258/TKI-258
54 nM
Sunitinib
5.5 nM
VX-680/MK-0457
65 nM