BLK
KINASE INFORMATION
Kinase Name
B lymphoid tyrosine kinase
Entrez Gene Symbol
BLK
Entrez Gene ID
640
Aliases
BLK; MGC10442
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_001706.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.76
Panel
Delta Set M; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AST-487
30 nM
Dasatinib
0.21 nM
Sunitinib
65 nM