BMPR2
KINASE INFORMATION
Kinase Name
bone morphogenetic protein receptor, type II (serine/threonine kinase)
Entrez Gene Symbol
BMPR2
Entrez Gene ID
659
Aliases
BMPR2; BMPR3; BMPR-II; BMR2; BRK-3; FLJ41585; FLJ76945; PPH1; T-ALK
Kinase Group
TKL
Species
Human
PROTEIN INFORMATION
Accession #
NP_001195.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.78
Panel
Delta Set CA; Delta Set CE; Delta Set I; Delta Set M; scanEDGE; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
1500 nM
JNJ-7706621
880 nM
SU-14813
200 nM