BRAF
KINASE INFORMATION
Kinase Name
v-raf murine sarcoma viral oncogene homolog B1
Entrez Gene Symbol
BRAF
Entrez Gene ID
673
Aliases
BRAF; BRAF1; B-RAF1; FLJ95109; MGC126806; MGC138284; RAFB1
Kinase Group
TKL
Species
Human
PROTEIN INFORMATION
Accession #
NP_004324.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.69
Panel
Delta Set M; scanEDGE; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AMG-706
630 nM
CHIR-265/RAF-265
1200 nM
Dasatinib
500 nM
Sorafenib
540 nM