BRK
KINASE INFORMATION
Kinase Name
protein tyrosine kinase 6
Entrez Gene Symbol
PTK6
Entrez Gene ID
5753
Aliases
BRK; FLJ42088; PTK6
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_005966.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.72
Panel
scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AMG-706
1000 nM
Dasatinib
7.8 nM
ZD-6474
160 nM