BRSK2
KINASE INFORMATION
Kinase Name
BR serine/threonine kinase 2
Entrez Gene Symbol
BRSK2
Entrez Gene ID
9024
Aliases
BRSK2; C11orf7; FLJ41362; PEN11B; SAD1; STK29
Kinase Group
CAMK
Species
Human
PROTEIN INFORMATION
Accession #
EAX02438.1
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.69
Panel
Delta Set CE; Delta Set I; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
16 nM
PKC-412
650 nM
Sunitinib
1100 nM