BTK
KINASE INFORMATION
Kinase Name
Bruton agammaglobulinemia tyrosine kinase
Entrez Gene Symbol
BTK
Entrez Gene ID
695
Aliases
AGMX1; AT; ATK; BPK; BTK; IMD1; MGC126261; MGC126262; PSCTK1; XLA
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_000052.1
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.69
Panel
scanEDGE; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
66 nM
Dasatinib
1.4 nM
Staurosporine
210 nM