CASK
KINASE INFORMATION
Kinase Name
calcium/calmodulin-dependent serine protein kinase (MAGUK family)
Entrez Gene Symbol
CASK
Entrez Gene ID
8573
Aliases
CAGH39; CAMGUK; CASK; CMG; FGS4; FLJ22219; FLJ31914; LIN2; MICPCH; TNRC8
Kinase Group
CAMK
Species
Human
PROTEIN INFORMATION
Accession #
NP_003679.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.75
Panel
Delta Set CA; Delta Set CE; Delta Set I; Delta Set M; Delta Set RB; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
K-252a
560 nM
Staurosporine
19 nM