CDK4-cyclinD3
KINASE INFORMATION
Kinase Name
cyclin-dependent kinase 4
Entrez Gene Symbol
CDK4
Entrez Gene ID
1019
Aliases
CDK4; CMM3; MGC14458; PSK-J3
Kinase Group
CMGC
Species
Human
PROTEIN INFORMATION
Accession #
NP_000066.1
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.7
Panel
scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
K-252a
6.4 nM
Purvalanol B
780 nM
Staurosporine
20 nM