CDK9
KINASE INFORMATION
Kinase Name
cyclin-dependent kinase 9
Entrez Gene Symbol
CDK9
Entrez Gene ID
1025
Aliases
C-2k; CDC2L4; CDK9; CTK1; PITALRE; TAK
Kinase Group
CMGC
Species
Human
PROTEIN INFORMATION
Accession #
NP_001252.1
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.72
Panel
scanEDGE; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
BMS-387032/SNS-032
76 nM
Flavopiridol
6.4 nM
JNJ-7706621
470 nM