CHEK2
KINASE INFORMATION
Kinase Name
CHK2 checkpoint homolog (S. pombe)
Entrez Gene Symbol
CHEK2
Entrez Gene ID
11200
Aliases
CDS1; CHEK2; CHK2; HuCds1; LFS2; PP1425; RAD53
Kinase Group
CAMK
Species
Human
PROTEIN INFORMATION
Accession #
NP_001005735.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.63
Panel
scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
210 nM
Staurosporine
74 nM
Sunitinib
7.1 nM