CIT
KINASE INFORMATION
Kinase Name
citron (rho-interacting, serine/threonine kinase 21)
Entrez Gene Symbol
CIT
Entrez Gene ID
11113
Aliases
CIT; CRIK; KIAA0949; STK21
Kinase Group
AGC
Species
Human
PROTEIN INFORMATION
Accession #
NP_009105.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.73
Panel
Delta Set I; Delta Set M; Delta Set RB; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AST-487
52 nM
CHIR-265/RAF-265
87 nM
Flavopiridol
110 nM