CSF1R
KINASE INFORMATION
Kinase Name
colony stimulating factor 1 receptor
Entrez Gene Symbol
CSF1R
Entrez Gene ID
1436
Aliases
CD115; C-FMS; CSF1R; CSF-1R; CSF-1-R; CSFR; FIM2; FIM-2; FMS; Fms/CSFR
Kinase Group
TK
Species
Human
Phosphorylated
yes
PROTEIN INFORMATION
Accession #
NP_005202.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.65
Panel
scanEDGE; scanELECT; scanMAX; scanMODE; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CHIR-258/TKI-258
60 nM
GW-2580
1.6 nM
MLN-518
4.9 nM
Pazopanib
7.9 nM
SU-14813
3.6 nM
Sunitinib
2 nM