CSK
KINASE INFORMATION
Kinase Name
c-src tyrosine kinase
Entrez Gene Symbol
CSK
Entrez Gene ID
1445
Aliases
CSK; MGC117393
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_004374.1
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.69
Panel
scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AST-487
2300 nM
CEP-701
260 nM
Dasatinib
1 nM