DDR2
KINASE INFORMATION
Kinase Name
discoidin domain receptor tyrosine kinase 2
Entrez Gene Symbol
DDR2
Entrez Gene ID
4921
Aliases
DDR2; MIG20a; NTRKR3; TKT; TYRO10
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
CAA52777.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.62
Panel
scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
Dasatinib
3.2 nM
Imatinib
15 nM
Sorafenib
6.6 nM