DLK
KINASE INFORMATION
Kinase Name
mitogen-activated protein kinase kinase kinase 12
Entrez Gene Symbol
MAP3K12
Entrez Gene ID
7786
Aliases
DLK; MAP3K12; MEKK12; MUK; ZPK; ZPKP1
Kinase Group
TKL
Species
Human
PROTEIN INFORMATION
Accession #
NP_006292.2
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.66
Panel
Delta Set I; Delta Set M; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
SU-14813
560 nM
Sunitinib
100 nM
VX-680/MK-0457
190 nM