DMPK
KINASE INFORMATION
Kinase Name
dystrophia myotonica-protein kinase
Entrez Gene Symbol
DMPK
Entrez Gene ID
1760
Aliases
DM; DM1; DM1PK; DMK; DMPK; MDPK; MT-PK
Kinase Group
AGC
Species
Human
PROTEIN INFORMATION
Accession #
NP_004400.4
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.62
Panel
Delta Set CA; Delta Set CE; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
240 nM
EKB-569
59 nM
Flavopiridol
650 nM