DRAK2
KINASE INFORMATION
Kinase Name
serine/threonine kinase 17b
Entrez Gene Symbol
STK17B
Entrez Gene ID
9262
Aliases
DRAK2; STK17B
Kinase Group
CAMK
Species
Human
PROTEIN INFORMATION
Accession #
NP_004217.1
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.57
Panel
Delta Set CA; Delta Set CE; Delta Set I; Delta Set M; Delta Set RB; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
MLN-8054
8.1 nM
SU-14813
320 nM
Sunitinib
110 nM