DYRK2
KINASE INFORMATION
Kinase Name
dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 2
Entrez Gene Symbol
DYRK2
Entrez Gene ID
8445
Aliases
DYRK2; FLJ21217; FLJ21365
Kinase Group
CMGC
Species
Human
PROTEIN INFORMATION
Accession #
NP_003574.1
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.71
Panel
Delta Set I; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
22 nM
Staurosporine
250 nM
Sunitinib
680 nM