ERBB4
KINASE INFORMATION
Kinase Name
v-erb-a erythroblastic leukemia viral oncogene homolog 4 (avian)
Entrez Gene Symbol
ERBB4
Entrez Gene ID
2066
Aliases
ERBB4; HER4; MGC138404; p180erbB4
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_001036064.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.72
Panel
scanEDGE; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CI-1033
29 nM
CP-724714
260 nM
EKB-569
21 nM
Gefitinib
410 nM
Lapatinib
54 nM