ERN1
KINASE INFORMATION
Kinase Name
endoplasmic reticulum to nucleus signaling 1
Entrez Gene Symbol
ERN1
Entrez Gene ID
2081
Aliases
ERN1; FLJ30999; hIRE1p; IRE1; IRE1a; IRE1P; MGC163277; MGC163279
Kinase Group
Other
Species
Human
PROTEIN INFORMATION
Accession #
NP_001424.3
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.55
Panel
Delta Set CA; Delta Set CE; Delta Set I; Delta Set M; Delta Set RB; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
PKC-412
2300 nM
Staurosporine
21 nM
Sunitinib
600 nM