FGFR3
KINASE INFORMATION
Kinase Name
fibroblast growth factor receptor 3
Entrez Gene Symbol
FGFR3
Entrez Gene ID
2261
Aliases
ACH; CD333; CEK2; FGFR3; HSFGFR3EX; JTK4
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_000133.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.76
Panel
scanEDGE; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
580 nM
CHIR-258/TKI-258
230 nM
Pazopanib
740 nM
SU-14813
560 nM
Sunitinib
290 nM