FGFR4
KINASE INFORMATION
Kinase Name
fibroblast growth factor receptor 4
Entrez Gene Symbol
FGFR4
Entrez Gene ID
2264
Aliases
CD334; FGFR4; JTK2; MGC20292; TKF
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_075252.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.62
Panel
scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AST-487
1400 nM
CEP-701
1800 nM
CHIR-258/TKI-258
4300 nM
Pazopanib
2800 nM