FGR
KINASE INFORMATION
Kinase Name
Gardner-Rasheed feline sarcoma viral (v-fgr) oncogene homolog
Entrez Gene Symbol
FGR
Entrez Gene ID
2268
Aliases
c-fgr; c-src2; FGR; FLJ43153; MGC75096; p55c-fgr; p55-Fgr; p58c-fgr; SRC2
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_005239.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.7
Panel
scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AST-487
190 nM
CEP-701
52 nM
Dasatinib
0.5 nM