FLT3
KINASE INFORMATION
Kinase Name
fms-related tyrosine kinase 3
Entrez Gene Symbol
FLT3
Entrez Gene ID
2322
Aliases
CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1
Kinase Group
TK
Species
Human
Phosphorylated
yes
PROTEIN INFORMATION
Accession #
NP_004110.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.7
Panel
scanEDGE; scanELECT; scanMAX; scanMODE; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
ABT-869
0.63 nM
CEP-701
8.5 nM
CHIR-258/TKI-258
0.64 nM
MLN-518
3 nM
PKC-412
11 nM
Sunitinib
0.47 nM