FLT4
KINASE INFORMATION
Kinase Name
fms-related tyrosine kinase 4
Entrez Gene Symbol
FLT4
Entrez Gene ID
2324
Aliases
FLT4; FLT41; LMPH1A; PCL; VEGFR3
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_002011.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.68
Panel
scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AMG-706
9.7 nM
CHIR-258/TKI-258
580 nM
Pazopanib
27 nM
SU-14813
50 nM
Sunitinib
50 nM
ZD-6474
1100 nM