GAK
KINASE INFORMATION
Kinase Name
cyclin G associated kinase
Entrez Gene Symbol
GAK
Entrez Gene ID
2580
Aliases
FLJ16629; FLJ40395; GAK; MGC99654
Kinase Group
Other
Species
Human
PROTEIN INFORMATION
Accession #
NP_005246.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.77
Panel
Delta Set CA; Delta Set CE; Delta Set I; Delta Set M; Delta Set RB; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
Erlotinib
3.1 nM
SB-203580
19 nM
SU-14813
44 nM