GCN2(Kin.Dom.2,S808G)
KINASE INFORMATION
Kinase Name
eukaryotic translation initiation factor 2 alpha kinase 4
Entrez Gene Symbol
EIF2AK4
Entrez Gene ID
440275
Aliases
EIF2AK4; GCN2; KIAA1338
Kinase Group
Other
Species
Human
PROTEIN INFORMATION
Accession #
NP_001013725.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.73
Panel
Delta Set CA; Delta Set CE; Delta Set I; Delta Set M; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CGP-52421
16 nM
CHIR-265/RAF-265
55 nM
PKC-412
39 nM