GRK7
KINASE INFORMATION
Kinase Name
G protein-coupled receptor kinase 7
Entrez Gene Symbol
GRK7
Entrez Gene ID
131890
Aliases
GPRK7; GRK7
Kinase Group
AGC
Species
Human
PROTEIN INFORMATION
Accession #
NP_631948.1
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.71
Panel
Delta Set CA; Delta Set CE; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
7.2 nM
PKC-412
48 nM
Sunitinib
180 nM