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IGF1R

KINASE INFORMATION

Kinase Name insulin-like growth factor 1 receptor
Entrez Gene Symbol IGF1R
Entrez Gene ID 3480
Aliases CD221; IGF1R; IGFIR; IGFR; JTK13; MGC142170; MGC142172; MGC18216
Kinase Group TK
Species Human

PROTEIN INFORMATION

Accession # NP_000866.1
Kinase Construct Partial Length
Kinase Form Wild Type
Expression System Bacterial

ASSAY INFORMATION

Average Z’ Value 0.63
Panel scanEDGE; scanELECT; scanMAX; scanTK;

REFERENCE INHIBITOR INFORMATION

CompoundKd
Staurosporine210 nM
Sunitinib2600 nM
VX-680/MK-0457740 nM

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