IKK-alpha
KINASE INFORMATION
Kinase Name
conserved helix-loop-helix ubiquitous kinase
Entrez Gene Symbol
CHUK
Entrez Gene ID
1147
Aliases
CHUK; IKBKA; IKK1; IKKA; IKKalpha; IKK-alpha; NFKBIKA; TCF16
Kinase Group
Other
Species
Human
PROTEIN INFORMATION
Accession #
NP_001269.3
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.72
Panel
scanEDGE; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
9 nM
PKC-412
3800 nM
Sunitinib
520 nM