IKK-epsilon
KINASE INFORMATION
Kinase Name
inhibitor of kappa light polypeptide gene enhancer in B-cells, kinase epsilon
Entrez Gene Symbol
IKBKE
Entrez Gene ID
9641
Aliases
IKBKE; IKKE; IKK-E; IKKepsilon; IKK-epsilon; IKKI; IKK-i; KIAA0151; MGC125294; MGC125295; MGC125297
Kinase Group
Other
Species
Human
PROTEIN INFORMATION
Accession #
NP_054721.1
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.63
Panel
Delta Set M; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
11 nM
PKC-412
160 nM
Staurosporine
5.1 nM