INSR
KINASE INFORMATION
Kinase Name
insulin receptor
Entrez Gene Symbol
INSR
Entrez Gene ID
3643
Aliases
CD220; HHF5; INSR; IR
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_000199.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.65
Panel
scanEDGE; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
Staurosporine
110 nM
Sunitinib
500 nM
VX-680/MK-0457
630 nM