ITK
KINASE INFORMATION
Kinase Name
IL2-inducible T-cell kinase
Entrez Gene Symbol
ITK
Entrez Gene ID
3702
Aliases
EMT; ITK; LYK; MGC126257; MGC126258; PSCTK2
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_005537.3
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.75
Panel
scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
SU-14813
190 nM
Sunitinib
13 nM
VX-680/MK-0457
350 nM