JAK1(JH1domain-catalytic)
KINASE INFORMATION
Kinase Name
Janus kinase 1
Entrez Gene Symbol
JAK1
Entrez Gene ID
3716
Aliases
JAK1; JAK1A; JAK1B; JAK1-catalytic; JTK3
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_002218.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.66
Panel
Delta Set M; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
8.8 nM
CGP-52421
4400 nM
PKC-412
670 nM