JAK1(JH2domain-pseudokinase)
KINASE INFORMATION
Kinase Name
Janus kinase 1
Entrez Gene Symbol
JAK1
Entrez Gene ID
3716
Aliases
JAK1; JAK1~b; JAK1A; JAK1B; JAK1-pseudokinase; JTK3
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_002218.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.79
Panel
Delta Set M; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
JNJ-7706621
21 nM
SU-14813
97 nM
Sunitinib
49 nM