JAK3(JH1domain-catalytic)
KINASE INFORMATION
Kinase Name
Janus kinase 3
Entrez Gene Symbol
JAK3
Entrez Gene ID
3718
Aliases
JAK3; JAK-3; JAK3_HUMAN; JAK3-catalytic; JAKL; LJAK; L-JAK
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_000206.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.74
Panel
scanEDGE; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CP-690550
2.2 nM
PKC-412
12 nM
VX-680/MK-0457
630 nM