KIT
KINASE INFORMATION
Kinase Name
v-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog
Entrez Gene Symbol
KIT
Entrez Gene ID
3815
Aliases
CD117; C-Kit; KIT; PBT; SCFR
Kinase Group
TK
Species
Human
Phosphorylated
yes
PROTEIN INFORMATION
Accession #
NP_000213.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.77
Panel
scanEDGE; scanELECT; scanMAX; scanMODE; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AMG-706
3.7 nM
AST-487
5.4 nM
Imatinib
14 nM
MLN-518
2.7 nM
PKC-412
220 nM
Sunitinib
0.37 nM