LCK
KINASE INFORMATION
Kinase Name
lymphocyte-specific protein tyrosine kinase
Entrez Gene Symbol
LCK
Entrez Gene ID
3932
Aliases
LCK; LSK; p56lck; pp58lck; YT16
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_005347.3
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.76
Panel
scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
Dasatinib
0.2 nM
Imatinib
40 nM
ZD-6474
17 nM