LKB1
KINASE INFORMATION
Kinase Name
serine/threonine kinase 11
Entrez Gene Symbol
STK11
Entrez Gene ID
6794
Aliases
LKB1; PJS; STK11
Kinase Group
CAMK
Species
Human
PROTEIN INFORMATION
Accession #
NP_000446.1
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.63
Panel
Delta Set CE; Delta Set I; scanEDGE; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
PKC-412
350 nM
SU-14813
360 nM
Sunitinib
38 nM