LOK
KINASE INFORMATION
Kinase Name
serine/threonine kinase 10
Entrez Gene Symbol
STK10
Entrez Gene ID
6793
Aliases
LOK; PRO2729; STK10
Kinase Group
STE
Species
Human
PROTEIN INFORMATION
Accession #
NP_005981.3
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.73
Panel
Delta Set CE; Delta Set I; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AST-487
0.92 nM
CHIR-265/RAF-265
60 nM
Sunitinib
19 nM