LRRK2
KINASE INFORMATION
Kinase Name
leucine-rich repeat kinase 2
Entrez Gene Symbol
LRRK2
Entrez Gene ID
120892
Aliases
AURA17; DARDARIN; LRRK2; PARK8; RIPK7; ROCO2
Kinase Group
TKL
Species
Human
PROTEIN INFORMATION
Accession #
NP_940980.3
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.73
Panel
Delta Set CA; Delta Set M; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
K-252a
3.4 nM
Purvalanol B
750 nM
Staurosporine
3.1 nM