LRRK2(G2019S)
KINASE INFORMATION
Kinase Name
leucine-rich repeat kinase 2
Entrez Gene Symbol
LRRK2
Entrez Gene ID
120892
Aliases
AURA17; DARDARIN; LRRK2; PARK8; RIPK7; ROCO2
Kinase Group
TKL
Species
Human
PROTEIN INFORMATION
Accession #
NP_940980.3
Kinase Construct
Partial Length
Kinase Form
Mutation (G2019S)
Mutation Relevance
Activating mutation found in Parkinson's disease.
Mutation References
Proc Natl Acad Sci USA.
102, 16842-16847 (2005)
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.76
Panel
scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
K-252a
1.8 nM
Purvalanol B
670 nM
Staurosporine
0.39 nM